Perhal AF, Papadopoulos MGE, Medel-Lacruz B, Ladurner A, Selent J, Dirsch V et al. Discovery and characterization of small-molecule TGR5 ligands with agonistic activity. European Journal of Medicinal Chemistry. 2024 Jun 28. doi: 10.1016/j.ejmech.2024.116616

Czollner L, Papaplioura E, Linder T, Liu R, Li Y, Atanasov AG et al. A silver-coated copper wire as inexpensive drug eluting stent model: determination of the relative releasing properties of leoligin and derivatives. Monatshefte fur Chemie. 2023 Dec;154(12):1317-1326. Epub 2020 Nov 5. doi: 10.1007/s00706-020-02677-4

He Z, Zhang Z, Xu P, Dirsch VM, Wang L, Wang K. Laminarin Reduces Cholesterol Uptake and NPC1L1 Protein Expression in High-Fat Diet (HFD)-Fed Mice. Marine Drugs. 2023 Dec;21(12):624. doi: 10.3390/md21120624

Resetar M, Tietcheu Galani BR, Tsamo AT, Chen Y, Schachner D, Stolzlechner S et al. Flindissone, a Limonoid Isolated from Trichilia prieuriana, Is an LXR Agonist. Journal of Natural Products. 2023 Aug 25;86(8):1901-1909. doi: 10.1021/acs.jnatprod.3c00059

Zwirchmayr J, Schachner D, Grienke U, Rudžionytė I, de Martin R, Dirsch VM et al. Biochemometry identifies suppressors of pro-inflammatory gene expression in Pterocarpus santalinus heartwood. Phytochemistry. 2023 Aug;212:113709. doi: 10.1016/j.phytochem.2023.113709

Cannavacciuolo C, Cerulli A, Dirsch VM, Heiss EH, Masullo M, Piacente S. LC-MS- and ¹H NMR-Based Metabolomics to Highlight the Impact of Extraction Solvents on Chemical Profile and Antioxidant Activity of Daikon Sprouts (Raphanus sativus L.). Antioxidants. 2023 Aug;12(8):1542. doi: 10.3390/antiox12081542

Lapinskaite R, Atalay HN, Malatinec Š, Donmez S, Cinar ZO, Schwarz P et al. Synthesis of Selagibenzophenone A and Its Derivatives for Evaluation of Their Antiproliferative, RORγ Inverse Agonistic, and Antimicrobial Effect. Chemistry SELECT. 2023 Feb 13;8(7).

Blažević T, Ciotu CI, Gold-Binder M, Heiss EH, Fischer MJM, Dirsch VM. Cultured rat aortic vascular smooth muscle cells do not express a functional TRPV1. PLoS ONE. 2023 Feb;18(2):e0281191. doi: 10.1371/journal.pone.0281191

Cannavacciuolo C, Napolitano A, Heiss EH, Dirsch VM, Piacente S. Portulaca oleracea, a rich source of polar lipids: Chemical profile by LC-ESI/LTQOrbitrap/MS/MSn and in vitro preliminary anti-inflammatory activity. Food Chemistry. 2022 Sept 15;388:132968. doi: 10.1016/j.foodchem.2022.132968

Schwarz P, Perhal A, Schöberl LN, Kraus MM, Kirchmair J, Dirsch V. Identification of the Natural Steroid Sapogenin Diosgenin as a Direct Dual-Specific RORα/γ Inverse Agonist. Biomedicines. 2022 Aug;10(9). doi: 10.3390/biomedicines10092076

Pferschy-Wenzig EM, Ortmann S, Atanasov AG, Hellauer K, Hartler J, Kunert O et al. Characterization of Constituents with Potential Anti-Inflammatory Activity in Chinese Lonicera Species by UHPLC-HRMS Based Metabolite Profiling. Metabolites. 2022 Apr;12(4):288. doi: 10.3390/metabo12040288

Linder T, Papaplioura E, Ogurlu D, Geyrhofer S, Hummelbrunner S, Schachner D et al. Investigation of Leoligin Derivatives as NF-κΒ Inhibitory Agents. Biomedicines. 2022 Jan;10(1):62. Epub 2021 Dec 28. doi: 10.3390/biomedicines10010062

Hou X, Malainer C, Atanasov AG, Heiß EH, Dirsch VM, Wang L et al. Evodiamine Lowers Blood Lipids by Up-Regulating the PPARγ/ABCG1 Pathway in High-Fat-Diet-Fed Mice. Journal of Natural Products. 2021 Dec 24;84(12):3110-3116. doi: 10.1021/acs.jnatprod.1c00881

Ladurner A, Schwarz P, Dirsch V. Natural products as modulators of retinoic acid receptor-related orphan receptors (RORs). Natural Product Reports - NPR. 2021 Apr;38(4):757-781. Epub 2020 Oct 29. doi: 10.1039/D0NP00047G

Atanasov AG, Zotchev SB, Dirsch VM, the International Natural Product Sciences Taskforce, Supuran CT. Natural products in drug discovery: advances and opportunities. Nature Reviews Drug Discovery. 2021 Mar;20:200-216. Epub 2021 Jan 28. doi: 10.1038/s41573-020-00114-z

Blažević T, Reznicek G, Ding L, Yang G, Haiss P, Heiss EH et al. Short Chain (≤C4) Esterification Increases Bioavailability of Rosmarinic Acid and Its Potency to Inhibit Vascular Smooth Muscle Cell Proliferation. Frontiers in Pharmacology. 2021 Jan 21;11:609756. doi: 10.3389/fphar.2020.609756

Ladurner A, Linder T, Wang L, Hiebl V, Schuster D, Schnürch M et al. Characterization of a structural leoligin analog as farnesoid X receptor agonist and modulator of cholesterol transport. Planta Medica. 2020 Oct 1;86(15):1097-1107. doi: 10.1055/a-1171-8357

Dao-Huy T, Latkolik S, Bräuer J, Pfeil A, Stuppner H, Schnürch M et al. Structural features defining nf-κb inhibition by lignan-inspired benzofurans and benzothiophenes. Biomolecules. 2020 Aug;10(8):1131. doi: 10.3390/biom10081131

Wang D, Hiebl V, Schachner D, Ladurner A, Heiss EH, Atanasov AG et al. Soraphen A enhances macrophage cholesterol efflux via indirect LXR activation and ABCA1 upregulation. Biochemical Pharmacology. 2020 Jul;177:114022. doi: 10.1016/j.bcp.2020.114022

Zwirchmayr J, Grienke U, Hummelbrunner S, Seigner J, de Martin R, Dirsch VM et al. A biochemometric approach for the identification of in vitro anti-inflammatory constituents in masterwort. Biomolecules. 2020 May;10(5):679. doi: 10.3390/biom10050679